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14 Cards in this Set
- Front
- Back
Substrates for CYP1A2
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Amitriptyline
Clomipramine Clozapine Desipramine Fluvoxamine Haloperidol Impramine Ropinirole Tacrine Theophylline (R)- Warfarin |
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Substrates for CYP2C9
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Diazepam
Phenytoin (S)- Warfarin |
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Substrates for CYP2C19
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Phenytoin
Thioridazine |
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Substrates for CYP2D6
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Amitriptyline
Atomoxetine Codeine Desipramine Dextromethorphan Donepezil Doxepin Fentanyl Flecainide Haloperidol Hydrocodone Imipramine Meperidine Methadone Mexiletine Nortriptyline Oxycodone Propafenone Propoxyphene Thioridazine Tramadol Trazodone |
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Inhibitors of CYP 1A2
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Cimetidine
Ciprofloxacin Clarithromycin Enoxacin Erythromycin Fluvoxamine Isoniazid Nalidixic acid Norfloxacin Troleandomycin Zileuton |
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Inducers of CYP 1A2
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Carbamazepine
Phenobarbital Phenytoin Primidone Rifampin Ritonavir Smoking St. John's wort |
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Inhibitors of CYP 2C9
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Amiodarone
Chloramphenicol Cimetidine Fluconazole Fluvoxamine Isoniazid Metronidazole Voriconazole Zafirlukast |
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Inducers of CYP 2C9
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Carbamazepine
Phenobarbital Phenytoin Primidone Rifampin Rifapentine |
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Inhibitors of CYP 2C19
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Fluoxetine
Fluvoxamine Modafinil Omeprazole Topiramate |
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Inducers of CYP 2C19
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Carbamazepine
Phenobarbital Phenytoin |
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Inhibitors of CYP 2D6
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Amiodarone
Cimetidine Fluoxetine Paroxetine Quinidine Ritonavir Sertraline |
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Inducers of CYP 2D6
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St. John's Wort
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Inhibitors of CYP 3A4
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Amiodarone
Cimetidine Ciprofloxacin Clarithromycin Cyclosporine Delavirdine Diltiazem Efavirenz Erythromycin Fluconazole Fluoxetine Fluvoxamine Grapefruit Indinavir Isoniazid Itraconazole Ketoconazole Metronidazole Miconazole Nefazodone Nelfinavir Nefedipine Norfloxacin Quinine Ritonavir |
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Inducers of CYP 3A4
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Carbamazepine
Efavirenz Ethosucimide Garlic supplements Modafinil Nevirapine Oxcarbazepine Phenobarbital Phenytoin Primidone Rifabutin Rifapentine St. John's Wort |