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134 Cards in this Set
- Front
- Back
Cimetidine
|
H2 Receptor Antagonist
|
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Ranitidine
|
H2 Receptor Antagonist
|
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Omeprazole
|
Proton Pump Inhibitor
|
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Pirenzepine
|
Muscarinic M1 Antagonist
(The Original Anti-Ulcer Drug) (Not used anymore due to side effects) |
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Aluminium Hydroxide
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Antacid
|
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Magnesium Hydroxide
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Antacid
|
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Sodium Bicarbonate
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Antacid
|
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Sucralfate
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Mucosal Protectant
|
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Colloidal Bismuth
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Mucosal Protectant
|
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Misoprostol
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Synthetic Prostaglandin E1 |
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Indomethacin
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Cyclooxygenase Inhibitor
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Ibuprophen
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Cyclooxygenase Inhibitor
|
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Colchicine
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Microtubule Assembly Inhibitor
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Allopurinol
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Competitive Xanthine Oxidase Inhibitor
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Probenecid
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Uricosuric Agent
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Sulphinpyrazone
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Uricosuric Agent
|
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Uricase
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Uric Acid Metabolizer
|
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Hydroxychloroquine
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Disease Modifying Antirheumatic Drug (DMARD)
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Sulphasalazine
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Disease Modifying Antirheumatic Drug (DMARD)
|
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Sodium Aurothiomalate
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Gold Salt
Macrophage Suppression |
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Aurofin
|
Gold Salt
Macrophage Suppression |
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Penicillamine
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Chelates Heavy Metals
|
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Methotraxate
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Folic Acid Antagonist
|
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Leflunomide
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Dihydroorotate Dehydrogenase Inhibitor
|
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Azathioprine
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Purine Analogue Cytotoxic to Inflammatory Cells
|
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Cyclosporine
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Antibiotic
|
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Salbutamol
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Beta 2 Agonist
|
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Adrenaline
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Non-Selective Adrenergic Agonist
|
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Isoprenaline
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Non-Selective Adrenergic Agonist
|
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Theophylline
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Phosphodiesterase Inhibitor
Xanthine Class |
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Ipratropium
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Non-Selective Muscarinic Receptor Antagonist
|
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Cromoglycate
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Prophylactic Agent for Asthmatics
|
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Beclomethasone
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Glucocorticoid
|
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Zileuton
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5-Lipoxygenase Inhibitor
|
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Zafirlukast
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cysLT1 Receptor Antagonist
|
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Montelukast
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cysLT1 Receptor Antagonist
|
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Nifedipine (Inhaled)
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Calcium Channel Blocker
|
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Verapamil (Inhaled)
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Calcium Channel Blocker
|
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Chromakalim
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Potassium Channel Openers
|
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Omalizumab
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Anti-IgE Monoclonal Antibodies
|
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Tropicamide
|
Muscarinic Antagonist
|
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Timolol
|
Beta Receptor Antagonist
|
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Dorzolamide
|
Carbonic Anhydrase Inhibitor
|
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Pilocarpine
|
Muscarinic Agonist
|
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Lanaprost
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Prostaglandin F2 alpha Analogue
|
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Verteprofin
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Photodynamic Therapy Agent
|
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Ranibizumab
|
VEGF Monoclonal Antibodies
|
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Metronidazole
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Prodrug of Cytotoxic, Antibiotic Compound
Clinically Used to Kill Amoeba and Anaerobic Organisms |
|
Pentamidine
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DHFR Inhibitor
Clinicallyused to treat Early Stage (non-CNS) in Trypanosomiasis (Sleeping Sickness) |
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Suramin
|
Multi-Enzyme Inhibitor
Clinicallyused to treat Early Stage (non-CNS) in Trypanosomiasis (Sleeping Sickness) |
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Melarsopol
|
Combination of Dimercaptopropanol and Melarsen Oxide (Arsenic Compound)
Clinicallyused to treat Late Stage (CNS) in Trypanosomiasis (Sleeping Sickness) |
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Sodium Stibogluconate
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Anti-Protazoal Agent
|
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Meglumine Antimonate
|
Anit-Protazoal Agent
|
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Miltefosine
|
Anti-Protazoal Agent
Synthetic Ether Phospholipid Analogue |
|
Ivermectin
|
Semisynthetic Macrocyclic Lactone
Clinically used against many Helminths and Arthropods |
|
Piperazine
|
GABA Receptor Agonist
Clinically used (historically) to treat Round Worm and Pin Worm |
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Pyrantel Pamoate
|
Cation Channel Agonist
Depolarizing Neuromuscular Blocking Agent Clinically Used as Third Line Agent against Hookworm, Pinworm, or Roundworm Infections |
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Albendazole
|
Microtubule Assembly Inhibitor
Anti-Helminthic Agent |
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Mebendazole
|
Microtuble Assembly Inhibitor
Anti-Helminthic Agent |
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Praziquantel
|
Anti-Helminthic Agent
|
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Diethylcarbamizine (DEC)
|
Piperazine Derivative
Anti-Helminthic Agent |
|
Erlotinib
|
EGFR Inhibitor
Anti-Cancer Agent |
|
Cetuximab
|
Chimeric Mouse/Human IgG1 Monoclonal Antibody to EGFR (ErbB1)
Anti-Cancer Agent |
|
Trastuzumab
|
Chimeric Mouse/Human IgG1 Monoclonal Antibody to EGFR (ErbB2)
Anti-Cancer Agent |
|
Imatinib Mesylate
|
Tyrosine Kinase Inhibitor
Anti-Cancer Agent |
|
Tipifarnib
|
Farnesyltransferase Inhibitor
Clinically used for Relapsed/Refractory AML |
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Sorafenib
|
Multiple rTK Inhibitor (VEGFR-1, VEGFR-2, PDGFR, and B-RAF Kinase)
Anti-Cancer Agent |
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Bortezomib
|
Proteasome Inhibitor
Anti-Cancer Agent |
|
Bevacizumab
|
Humanised Mouse IgG1 Antibody against VEGF-A
Anti-Cancer Agent |
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Vatalanib
|
VEGFR-1 and VEGFR-2 Inhibitor
|
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Rituximab
|
Anti-CD20 Antibody
Targets B Cell Non-Hodgkin's Lymphoma |
|
Alemtuzumab
|
Anti-CD52 Antibody
Targets Chronic Lymphocytic Leukaemia |
|
Gemtuzumab
|
Anti-CD33 Antibody Conjugated to Calicheamicin
Targets Acute Myeloid Leukaemia |
|
Enfuvirtide
|
Anti-HIV Peptide
Fusion Inhibitor Anti-HIV Drrug |
|
Amantadine
|
Ion Channel Inhibitor
Anti-Influenza A Drug |
|
Rimantadine
|
Ion Channel Inhibitor
Anti-Influenza A Drug |
|
Raltegravir
|
HIV Integrase Inhibitor
Anti-HIV Drug |
|
Zidovudine (AZT)
|
Thymidine Analogue
Nucleoside Reverse Transcriptase Inhibitor (NRTI) Anti-HIV Drug |
|
Lamivudine (3TC)
|
Cytidine Analogue
Nucleoside Reverse Transciptase Inhibitor (NRTI) Anti-HIV Drug |
|
Acyclovir
|
Guanine Base Attached to Incomplete Sugar
Anti-HSV/VCZ Drug |
|
Efavirenz
|
Non-Nucleoside Reverse Transcriptase Inhibitor (NNRTI)
Anti-HIV Drug |
|
Nevirapine
|
Non-Nucleoside Reverse Transcriptase Inhibitor (NNRTI)
Anti-HIV Drug |
|
Ritonavir
|
HIV Protease Inhibitor
Anti-HIV Drug |
|
Saquinavir
|
HIV Protease Inhibitor
Anti-HIV Drug |
|
Zanamivir
|
Sialic Acid Analogue
Anti-Influenza Drug |
|
Oseltamivir
|
Prodrug Sialic Acid Analogue
Anti-Influenza Drug |
|
Ketoconazole
|
CYP450 Enzyme Inhibitor (specifically ones involved with production of Cortisol and Aldosterone) |
|
Metyrapone
|
Reversible 11 beta - Hyroxylase Inhibitor
|
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Hydrocortisone (Cortisol)
|
Endogenous Glucocorticoid
|
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Cortisone
|
Pro-Drug Version of Glucocorticoid
|
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Prednisone
|
Pro-Drug Version of Glucocorticoid
|
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Prednisolone
|
Synthetic Glucocorticoid
|
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Dexamethasone
|
Synthetic Glucocorticoid
|
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Fluticasone
|
Synthetic Glucocorticoid
|
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Beclomethasone
|
Synthetic Glucocorticoid
|
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Methylprednisolone
|
Synthetic Cortisol Analogue
|
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Fludrocortisone
|
Synthetic Cortisol Analogue with High Mineralocorticoid Activity
|
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Spironolactone
|
Competative Aldosterone Receptor Antagonist
Potassium Sparing Diuretic |
|
Eplerenone
|
Competitve Aldosterone Receptor Antagonist
Potassium Sparing Diuretic |
|
Simvastatin
|
HMG-CoA Reductase Inhibitor
(Reversible and Competitive) Short Acting Statin |
|
Lovastatin
|
HMG-CoA Reductase Inhibitor
(Reversible and Competitive) Short Acting Statin |
|
Pravastatin
|
HMG-CoA Reductase Inhibitor
(Reversible and Competitive) Short Acting Statin |
|
Atorvastatin
|
HMG-CoA Reductase Inhibitor
(Reversible and Competitive) Long Acting Statin |
|
Rosuvastatin
|
HMG-CoA Reductase Inhibitor
(Reversible and Competitive) Long Acting Statin |
|
Gemfibrozil
|
Peroxisome Proliferator Activated Receptor Alpha (PPAR-alpha) Agonist
Fibrate Lipid Lowering Agent |
|
Fenofibrate
|
Peroxisome Proliferator Activated Receptor Alpha (PPAR-alpha) Agonist
Fibrate Lipid Lowering Agent |
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Ciprofibrate
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Peroxisome Proliferator Activated Receptor Alpha (PPAR-alpha) Agonist
Fibrate Lipid Lower Agent |
|
Colestyramine
|
Bile Acid-Binding Resin
Lipid Lowering Agent |
|
Colestipol
|
Bile Acid-Binding Resin
Lipid Lowering Agent |
|
Ezetimibe
|
Niemann-Pick C1-like 1 (NCPC1L1) Cholesterol Transport Protein Inhibitor
Cholesterol Absorption Inhibitor |
|
Niacin
|
Nicotinic Acid (Vitamin B3)
Lipid Lowering Agent |
|
Omacor
|
Polyunsaturated Fatty Acids
(Ex. Eicosapentaenoic and Docosahexaenoic Acid) Fish Oil Derivative Lipid Lowering Agent |
|
Aspirin
|
Irreversible Cyclooxygenase Inhibitor
First Line Anti-Platelet Agent |
|
Clopidogrel
|
Irreversible ADP Receptor Inhibitor
Second Line Anti-Platelet Agent (or combo with Aspirin) |
|
Prasugrel
|
Irreversible ADP Receptor Inhibitor
Anti-Platelet Agent |
|
Dipyridamole
|
Phosphodiesterase Inhibitor
Anti-Platelet Agent (relatively weak) |
|
Abciximab
|
Irreversible GPIIb-IIIa Antagonist (monoclonal antibody)
Anti-Platelet Agent |
|
Eptifibatide
|
GPIIb-IIIa Antagonist
|
|
Tirofiban
|
GPIIb-IIIa Antagonist
|
|
Heparin (unfractionated)
|
Thrombin and Factor Xa Inhibitor
Anti-Coagulant |
|
Dalteparin
|
Factor Xa Inhibitor
Anti-Coagulant Heparin (low molecular weight) |
|
Enoxaparin
|
Factor Xa Inhibitor
Anti-Coagulant Heparin (low molecular weight) |
|
Lepirudin
|
Direct Thrombin Inhibitor
|
|
Warfarin
|
Competitive Vitamin K Epoxide Reductase Component 1 (VKORC1) Inhibitor
Anti-Coagulant |
|
Dabigatran
|
Direct Thrombin Inhibitor
|
|
Rivaroxaban
|
Factor Xa Inhibitor
|
|
Protamine Sulphate
|
Heparin Antidote
|
|
Streptokinase
|
Plasminogen Activator
Fibrinolysis/Thrombolytic Agent |
|
Alteplase
|
Recombinant Tissue Plasminogen Activator (t-PA)
Fibrinolysis/Thrombolytic Agent |
|
Tranexamic Acid
|
Lysine Analogue
Plasminogen Activation Inhibitor Anti-Fibrinolytic Drugs |
|
Aminocaproic Acid
|
Lysine Analogue
Plasminogen Activation Inhibitor Anti-Fibrinolytic Drugs |
|
Desmopressin
|
Synthetic ADH Analogue
Anti-Fibrinolytic Drugs |
|
Etamyslate
|
Synthetic Haemostasis Drug
Indicated for short-term blood loss in menorrhagia |
|
Eptacog Alfa
|
Recombinant Factor VIIa
|