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99 Cards in this Set

  • Front
  • Back
Labetalol
alpha 1, beta 1/2 blocker
Carvediol
alpha 1, beta 1/2 blocker
Bucindolol
alpha 1, beta 1/2 blocker
Methyldopa
alpha 2 agonist, CNS
Clonidine
alpha 2 agonist, CNS
Hydrochlorothiazide
thiazide diuretic, "-azide"
Bendroflumethiazide
thiazide diuretic, "-azide"
Furosemide
loop diuretic, "-mide" or "-nide", sulfonamide derived
Indapamide
thiazide diuretic, "-azide"
Chlorothalidone
thiazide diuretic, "-azide"
Metolazone
thiazide diuretic, "-azide"
Chlorothiazide
thiazide diuretic, "-azide"
Methyclothiazide
thiazide diuretic, "-azide"
Tosemide
loop diuretic, "-mide" or "-nide", sulfonamide derived.
Polythiazide
thiazide diuretic, "-azide"
Trichloromethiazide
thiazide diuretic, "-azide"
Bumetanide
loop diuretic, "-mide" or "-nide", sulfonamide derived
Ethacrynic Acid
loop diuretic, non-sulfanamide, ototoxicity
Triameterne
K sparing, ENaC blocking
Amiloride
K sparing, ENaC blocking
Spirolactone
K sparing, Aldosterone blocking
Eplerenone
K sparing, Aldosterone blocking
Propranolol
non-specific beta blocker
Nadolol
non-specific beta blocker
Timolol
non-specific beta blocker
Pindolol
non-specific beta blocker
Carteolol
non-specific beta blocker
Levobunolol
non-specific beta blocker
Metoprolol
beta 1 specific beta blocker, "BEAM" blockers
Atenolol
beta 1 specific beta blocker, "BEAM" blockers
Betaxolol
beta 1 specific beta blocker, "BEAM" blockers
Bisoprolol
beta 1 specific beta blocker, "BEAM" blockers
Esmolol
beta 1 specific beta blocker, "BEAM" blockers
Acebutolol
beta 1 specific beta blocker, "BEAM" blockers
Nebivolol
biphasic beta blocker, <10mg B1 only, >10mg B1 &2, stimulate endothelial NO activity
Verapamil
non-Dihydropyridine (DHP) calcium channel blocker, works on heart and arterial vessels
Diltiazem
non-Dihydropyridine (DHP) calcium channel blocker, works on heart and arterial vessels
Nifedipine
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
Amlodipine
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
Isradipine
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
Felodipine
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
Nisoldipine
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
Nimodipine
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
Nicardipine
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
Clevidipine
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
Captopril
ACE inhibitor, "-pril"
Enalapril
ACE inhibitor, "-pril"
Lisinopril
ACE inhibitor, "-pril"
Ramipril
ACE inhibitor, "-pril"
Quinapril
ACE inhibitor, "-pril"
Fosinopril
ACE inhibitor, "-pril"
Benazepril
ACE inhibitor, "-pril"
Moexipril
ACE inhibitor, "-pril"
Perindopril
ACE inhibitor, "-pril"
Trandolapril
ACE inhibitor, "-pril"
Losartan
angiotensin II receptor blocker (ARB), "-sartan"
Valsartan
angiotensin II receptor blocker (ARB), "-sartan"
Candesartan
angiotensin II receptor blocker (ARB), "-sartan"
Irbesartan
angiotensin II receptor blocker (ARB), "-sartan"
Telmisartan
angiotensin II receptor blocker (ARB), "-sartan"
Eprosartan
angiotensin II receptor blocker (ARB), "-sartan"
Olmesartan
angiotensin II receptor blocker (ARB), "-sartan"
Aliskiren
Renin blocker
Phentolamine
non-specific alpha blocker, used in pheochromocytoma
Phenoxybenzamine
non-specific alpha blocker, used in pheochromocytoma
Prazosin
specific alpha 1 blocker, "-zosin"
Terazosin
specific alpha 1 blocker, "-zosin"
Doxazosin
specific alpha 1 blocker, "-zosin"
Mannatol
osmotic diuretic
Hydralazine
direct arterial vasodilator, MOA unknown
Minoxidil
direct arterial vasodilator, actives K channels on smooth muscle = hyper-polarization
Fenoldopam
activated D1 receptors on peripheral arteries (dilate) and renal artery (dilate)
Nitroprusside
dilate arteries and veins, NO cleaved at physiologic pH, NO activates cGMP (vasodilate)
Acetazolamide
carbonic anhydrase inhibitor, "-zolamide"
Brinzolamide
carbonic anhydrase inhibitor, "-zolamide"
Lovostatin
HMG CoA Reductase inhibitor, "-statin"
Fluvastatin
HMG CoA Reductase inhibitor, "-statin"
Pitavstatin
HMG CoA Reductase inhibitor, "-statin"
Pravastatin
HMG CoA Reductase inhibitor, "-statin"
Simvastatin
HMG CoA Reductase inhibitor, "-statin"
Atorvastatin
HMG CoA Reductase inhibitor, "-statin"
Rosuvastatin
HMG CoA Reductase inhibitor, "-statin"
Cerivastatin
HMG CoA Reductase inhibitor, "-statin"
Colesevelam
Bile acid binding resin
Colestipol
Bile acid binding resin
Cholestyramine
Bile acid binding resin
Niacin
block hormone sensitive lipase (HSL) in adipocytes (via GRP109A receptor) = decrease FFA release, block TG synthesis in liver (via blocking DGAT2), indirect breakdown of ApoB in liver
Ezetimibe
Block cholesterol absorption in enterocytes (NPC1L1 receptor blocker)
Sildenafil
Viagra, "-afil"
Vardenafil
Levetra, "-afil"
Tadalafil
Cialis, "-afil"
Gemfibrozil
Fibric acid derivative, activates PPAR-alpha to increase extra hepatic VLDL clearance, INCREASED RISK of rhabdomyolysis in combo with statin
Fenofibrate
Fibric acid derivative, activates PPAR-alpha to increase extra hepatic VLDL clearance
Finofibritic acid
Fibric acid derivative, activates PPAR-alpha to increase extra hepatic VLDL clearance
Amyl nitrate
vasodilate veins more then arteries (enzymes in venous walls free NO), work via NO cGMP, arterial dilation at high doses
Nitroglycerine
vasodilate veins more then arteries (enzymes in venous walls free NO), work via NO cGMP, arterial dilation at high doses
Isosorbide dinitrate
vasodilate veins more then arteries (enzymes in venous walls free NO), work via NO cGMP, arterial dilation at high doses
Isosorbide mononitrate
vasodilate veins more then arteries (enzymes in venous walls free NO), work via NO cGMP, arterial dilation at high doses
Ranolazine
block late I Na channels in myocytes