Use LEFT and RIGHT arrow keys to navigate between flashcards;
Use UP and DOWN arrow keys to flip the card;
H to show hint;
A reads text to speech;
99 Cards in this Set
- Front
- Back
Labetalol
|
alpha 1, beta 1/2 blocker
|
|
Carvediol
|
alpha 1, beta 1/2 blocker
|
|
Bucindolol
|
alpha 1, beta 1/2 blocker
|
|
Methyldopa
|
alpha 2 agonist, CNS
|
|
Clonidine
|
alpha 2 agonist, CNS
|
|
Hydrochlorothiazide
|
thiazide diuretic, "-azide"
|
|
Bendroflumethiazide
|
thiazide diuretic, "-azide"
|
|
Furosemide
|
loop diuretic, "-mide" or "-nide", sulfonamide derived
|
|
Indapamide
|
thiazide diuretic, "-azide"
|
|
Chlorothalidone
|
thiazide diuretic, "-azide"
|
|
Metolazone
|
thiazide diuretic, "-azide"
|
|
Chlorothiazide
|
thiazide diuretic, "-azide"
|
|
Methyclothiazide
|
thiazide diuretic, "-azide"
|
|
Tosemide
|
loop diuretic, "-mide" or "-nide", sulfonamide derived.
|
|
Polythiazide
|
thiazide diuretic, "-azide"
|
|
Trichloromethiazide
|
thiazide diuretic, "-azide"
|
|
Bumetanide
|
loop diuretic, "-mide" or "-nide", sulfonamide derived
|
|
Ethacrynic Acid
|
loop diuretic, non-sulfanamide, ototoxicity
|
|
Triameterne
|
K sparing, ENaC blocking
|
|
Amiloride
|
K sparing, ENaC blocking
|
|
Spirolactone
|
K sparing, Aldosterone blocking
|
|
Eplerenone
|
K sparing, Aldosterone blocking
|
|
Propranolol
|
non-specific beta blocker
|
|
Nadolol
|
non-specific beta blocker
|
|
Timolol
|
non-specific beta blocker
|
|
Pindolol
|
non-specific beta blocker
|
|
Carteolol
|
non-specific beta blocker
|
|
Levobunolol
|
non-specific beta blocker
|
|
Metoprolol
|
beta 1 specific beta blocker, "BEAM" blockers
|
|
Atenolol
|
beta 1 specific beta blocker, "BEAM" blockers
|
|
Betaxolol
|
beta 1 specific beta blocker, "BEAM" blockers
|
|
Bisoprolol
|
beta 1 specific beta blocker, "BEAM" blockers
|
|
Esmolol
|
beta 1 specific beta blocker, "BEAM" blockers
|
|
Acebutolol
|
beta 1 specific beta blocker, "BEAM" blockers
|
|
Nebivolol
|
biphasic beta blocker, <10mg B1 only, >10mg B1 &2, stimulate endothelial NO activity
|
|
Verapamil
|
non-Dihydropyridine (DHP) calcium channel blocker, works on heart and arterial vessels
|
|
Diltiazem
|
non-Dihydropyridine (DHP) calcium channel blocker, works on heart and arterial vessels
|
|
Nifedipine
|
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
|
|
Amlodipine
|
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
|
|
Isradipine
|
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
|
|
Felodipine
|
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
|
|
Nisoldipine
|
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
|
|
Nimodipine
|
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
|
|
Nicardipine
|
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
|
|
Clevidipine
|
Dihydropyridine (DHP) calcium channel blocker, arterial vessels only, "-dipine"
|
|
Captopril
|
ACE inhibitor, "-pril"
|
|
Enalapril
|
ACE inhibitor, "-pril"
|
|
Lisinopril
|
ACE inhibitor, "-pril"
|
|
Ramipril
|
ACE inhibitor, "-pril"
|
|
Quinapril
|
ACE inhibitor, "-pril"
|
|
Fosinopril
|
ACE inhibitor, "-pril"
|
|
Benazepril
|
ACE inhibitor, "-pril"
|
|
Moexipril
|
ACE inhibitor, "-pril"
|
|
Perindopril
|
ACE inhibitor, "-pril"
|
|
Trandolapril
|
ACE inhibitor, "-pril"
|
|
Losartan
|
angiotensin II receptor blocker (ARB), "-sartan"
|
|
Valsartan
|
angiotensin II receptor blocker (ARB), "-sartan"
|
|
Candesartan
|
angiotensin II receptor blocker (ARB), "-sartan"
|
|
Irbesartan
|
angiotensin II receptor blocker (ARB), "-sartan"
|
|
Telmisartan
|
angiotensin II receptor blocker (ARB), "-sartan"
|
|
Eprosartan
|
angiotensin II receptor blocker (ARB), "-sartan"
|
|
Olmesartan
|
angiotensin II receptor blocker (ARB), "-sartan"
|
|
Aliskiren
|
Renin blocker
|
|
Phentolamine
|
non-specific alpha blocker, used in pheochromocytoma
|
|
Phenoxybenzamine
|
non-specific alpha blocker, used in pheochromocytoma
|
|
Prazosin
|
specific alpha 1 blocker, "-zosin"
|
|
Terazosin
|
specific alpha 1 blocker, "-zosin"
|
|
Doxazosin
|
specific alpha 1 blocker, "-zosin"
|
|
Mannatol
|
osmotic diuretic
|
|
Hydralazine
|
direct arterial vasodilator, MOA unknown
|
|
Minoxidil
|
direct arterial vasodilator, actives K channels on smooth muscle = hyper-polarization
|
|
Fenoldopam
|
activated D1 receptors on peripheral arteries (dilate) and renal artery (dilate)
|
|
Nitroprusside
|
dilate arteries and veins, NO cleaved at physiologic pH, NO activates cGMP (vasodilate)
|
|
Acetazolamide
|
carbonic anhydrase inhibitor, "-zolamide"
|
|
Brinzolamide
|
carbonic anhydrase inhibitor, "-zolamide"
|
|
Lovostatin
|
HMG CoA Reductase inhibitor, "-statin"
|
|
Fluvastatin
|
HMG CoA Reductase inhibitor, "-statin"
|
|
Pitavstatin
|
HMG CoA Reductase inhibitor, "-statin"
|
|
Pravastatin
|
HMG CoA Reductase inhibitor, "-statin"
|
|
Simvastatin
|
HMG CoA Reductase inhibitor, "-statin"
|
|
Atorvastatin
|
HMG CoA Reductase inhibitor, "-statin"
|
|
Rosuvastatin
|
HMG CoA Reductase inhibitor, "-statin"
|
|
Cerivastatin
|
HMG CoA Reductase inhibitor, "-statin"
|
|
Colesevelam
|
Bile acid binding resin
|
|
Colestipol
|
Bile acid binding resin
|
|
Cholestyramine
|
Bile acid binding resin
|
|
Niacin
|
block hormone sensitive lipase (HSL) in adipocytes (via GRP109A receptor) = decrease FFA release, block TG synthesis in liver (via blocking DGAT2), indirect breakdown of ApoB in liver
|
|
Ezetimibe
|
Block cholesterol absorption in enterocytes (NPC1L1 receptor blocker)
|
|
Sildenafil
|
Viagra, "-afil"
|
|
Vardenafil
|
Levetra, "-afil"
|
|
Tadalafil
|
Cialis, "-afil"
|
|
Gemfibrozil
|
Fibric acid derivative, activates PPAR-alpha to increase extra hepatic VLDL clearance, INCREASED RISK of rhabdomyolysis in combo with statin
|
|
Fenofibrate
|
Fibric acid derivative, activates PPAR-alpha to increase extra hepatic VLDL clearance
|
|
Finofibritic acid
|
Fibric acid derivative, activates PPAR-alpha to increase extra hepatic VLDL clearance
|
|
Amyl nitrate
|
vasodilate veins more then arteries (enzymes in venous walls free NO), work via NO cGMP, arterial dilation at high doses
|
|
Nitroglycerine
|
vasodilate veins more then arteries (enzymes in venous walls free NO), work via NO cGMP, arterial dilation at high doses
|
|
Isosorbide dinitrate
|
vasodilate veins more then arteries (enzymes in venous walls free NO), work via NO cGMP, arterial dilation at high doses
|
|
Isosorbide mononitrate
|
vasodilate veins more then arteries (enzymes in venous walls free NO), work via NO cGMP, arterial dilation at high doses
|
|
Ranolazine
|
block late I Na channels in myocytes
|