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23 Cards in this Set
- Front
- Back
CHOLINERGIC AGONIST
WHAT ARE CHOLINE ESTERS DRUGS? |
BETHANECHOL (DUVOID)
TREATMENT OF BLADDER & GI HYPOTONIA |
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CHOLINERGIC AGONIST
WHAT ARE THE NEW M3 SPECIFIC AGONISTS DRUGS? |
CEVIMELINE (EVOXAC)
TREATMENT OF DRY MOUTH IN PTS WITH SJOGRENS SYNDROME |
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CHOLINERGIC AGONIST
WHAT ARE THE NATURAL ALKALOID DRUGS? |
PILOCARPINE (OCUSERT) (PILOCAR)
TREATMENT OF GLAUCOMA, TREAT DRY MOUTH (XEROSTOMIA) |
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In what areas of the body can AChE Inhibitors function on?
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All Autonomic Ganglia, Neuromuscular Junction, Eye, GI, Urinary Bladder, & effector organs innervated by PSNS.
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TYPES OF AChE INHIBITORS
What are the Reversible/Short drugs? |
EDROPHONIUM
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TYPES OF AChE INHIBITORS
What are the Reversible/Intermediate drugs? |
PHYSOSTIGMINE
NEOSTIGMINE PYRIDOSTIGMINE RIVASTIGMINE AMBENONIUM DONEPREZIL TACRINE |
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TYPES OF AChE INHIBITORS
What are the Irreversible/Synthetic Organophosphate drugs? |
ECOTHIOPHATE
ISOFLUOROPHATE (ECOTHIO- ISOFLUORO-) |
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TYPES OF AChE INHIBITORS
What are the Irreversible/Nerve Gases? |
SARIN
SOMA (SS) |
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WHAT ARE THE CLINICAL USES OF AChE INHIBITORS?
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TREATMENT OF:
-MYASTHENIA GRAVIS -HYPOTONIA OF BLADDER & GI -GLAUCOMA ALZHEIMERS |
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WHAT IS THE AChE INHIBITOR FIRST LINE OF DRUG AGAINST CHRONIC CASES/MYASTHENIA GRAVIS?
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NEOSTIGMINE
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WHAT ARE THE CLINICAL USES OF PHYSOSTIGMINE?
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-ANTIDOTE FOR OVERDOSES OF ATROPINE & ANTICHOLINERGIC DRUGS TO REVERSE CNS SIDE EFFECTS
-REDUCE IOP IN GLAUCOMA |
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WHAT ARE THE TREATMENTS FOR ORGANOPHOSPHATE/NERVE GAS POISONING?
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-PYRIDOSTIGMINE: PROPHYLACTICALLY IN CHEMICAL WARFARE
-POST EXPOSURE, HIGH DOSES OF MUSCARINIC ANTAGONIST ATROPINE OR SCOPOLAMINE FOLLOWED BY PRALIDOXIME (BEFORE AGING HAS OCCURRED) |
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MUSCARINIC RECEPTOR ANATAGONISTS
WHAT ARE THE BELLADONA ALKALOID DRUGS? |
-ATROPINE
-SCOPOLAMINE A.S. |
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MUSCARINIC RECEPTOR ANATAGONISTS
WHAT ARE THE SYNTHETIC & SEMI-SYNTHETIC DERIVATIVE DRUGS? |
-IPRATROPIUM
-TIOTROPIUM -TOLTERODINE T.I.T. |
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WHAT ARE THE SIDE EFFECTS OF ATROPINE?
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-DRY MOUTH
-CONSTIPATION -CYCLOPLEGIA (BLURRED VISION) -MYDRIASIS (DILATED PUPILS) -HOT, DRY FLUSHED SKIN -TACHYCARDIA -FEVER -CNS DISTURBANCES (ALL DOSAGE DEPENDANT) |
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WHAT ARE THE CLINICAL USES FOR SCOPOLAMINE?
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-PROPHYLACTIC FOR MOTION SICKNESS
-OPTHALMIC USE -ADJUNCT DRUG IN ANESTHESIA TO PRODUCE SEDATION & AMNESIA |
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WHAT ARE THE CLINICAL USES OF IPRATROPIUM BROMIDE (ATROVENT)?
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-CAUSE BRONCHODILATION AS AN ADJUNCT TO ALBUTEROL FOR ASTHMA & COPD PTS.
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WHAT ARE THE CLINICAL USES FOR TIOTROPIUM BROMIDE (SPIRIVA)?
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TREATMENT FOR COPD & ASTHMA
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WHAT ARE THE CLINICAL USES OF TOLTERODINE (DETROL)?
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TREATMENT OF OVERACTIVE BLADDER BY BLOCKING M3 RECEPTORS ON DETRUSOR MUSCLE REDUCING PSNS CONTRACTION OF BLADDER & DIMINISH URGE INCONTINENCE DURING FILLING
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NAME THE M3 ANTAGONISTS THAT ARE SIMILAR TO TOLTERODINE?
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-FESOTERODINE
-SOLIFENACIN -DARIFENACIN -OXYBUTYNIN |
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WHAT ARE THE CLINICAL USES FOR NEUROMUSCULAR JUNCTION BLOCKERS?
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SKELETAL MUSCLE RELAXANTS, USED IN SURGERY AS ADJUNCTS TO ANESTHESIA
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NMJ BLOCKERS
WHAT ARE THE NON-DEPOLORIZING BLOCKER DRUGS |
-ATRACURIUM
-CISTRACURIUM -VECURONIUM -ROCURONIUM -PANCURONIUM -TUBOCURARINE |
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NMJ BLOCKERS
WHAT ARE THE DEPOLARIZING DRUGS? |
SUCCINYL CHOLINE
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