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42 Cards in this Set

  • Front
  • Back
Norepinephrine
"short duration (broken down by COMT+MAO)
Epinephrine
"short duration (broken down by COMT+MAO)
Isoproterenol
"long duration (broken down by COMT, but not MAO)
phenylephrine
"a1-agonist
clonidine
"a2 agonist
apraclonidine
"a2-agonist
brimonidine
"a2-agonist
dobutamine
"b1-agonist
terbutaline
"b2-agonist
albuterol
"b2-agonist
Amphetamine
"a, b,CNS - agonist
Epedrine, Pseudoepedrine
"a, b,CNS - agonist
Reserpine
blocks NE vesicle transport
Tyramine
displacement of NE transmitter (axon terminal), causes increase release and increases flight or flight response
Cocaine
"inhibits NE reuptake
Phenoxybenzamine
"a-nonselective-BLOCKER
Phentolamine
"a-nonselective-BLOCKER
Prazosin
"a1-Antagonist
Dapiprazole
"a1-antagonist
yohimbine
"a2-antagonist
Propanolol
"nonselective B-blocker
Timolol
"nonselective B-blocker
Metoprolol
"B1-Blocker (cardioselective)
Esmolol
"B1-blocker (cardio selective)
Carvedilol
"a1,b1,b2-blocker (3rd gen, nonselective b-blocker w/ vasodilation)
a-methyl tyrosine
inhibits neurotransmitter sythesis
Methyldopa
alters dopamine function
guanadrel, Bretylium
inhibits release of NE
Acetylcholine
"Muscarinic agonists (direct cholinomimetics)
Bethanecol
"Muscarinic agonists (direct cholinomimetics)
Pilocarpine
"Muscarinic agonists (direct cholinomimetics)
Edrophonium
"Reversible acetylcholinesterase inhibitors (indirect-acting cholinomimetics)
Neostigmine
"Reversible acetylcholinesterase inhibitors (indirect-acting cholinomimetics)
Physostigmine
"Reversible acetylcholinesterase inhibitors (indirect-acting cholinomimetics)
Echothiophate
"Irreversible acetylcholinesterase inhibitors (indirect-acting cholinomimetics)
Isoflurophate (DFP)
"Irreversible acetylcholinesterase inhibitors (indirect-acting cholinomimetics)
Pralidoxime (2-PAM)
"acetylcholinesterase inhibitors (indirect-acting cholinomimetics)
Atropine
"Muscarinic Antagonist (cholinerigic antagonist)
Ipratropium
"Muscarinic Antagonist (cholinerigic antagonist)
Scopolamine
"Muscarininc Antagonist (cholinerigic antagonist)
Tropicamide
"Muscarinic antagonist (cholinerigic antagonist)
Cyclopentolate
"Muscarinic antagonist (cholinerigic antagonist)